Slow, tight-binding inhibition of PDF by actinonin induces

Inhibition and enzymatic reactions progress through an induced fit

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A [(32)P]NAD(+)-based method to identify and quantitate long residence time enoyl-acyl carrier protein reductase inhibitors. - Abstract - Europe PMC

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Slow, tight-binding inhibition of PDF by actinonin induces

3D comparison of the binding between various PDFIs and actinonin.: (a)

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Michel Desmadril's research works Université Paris-Saclay, Paris and other places

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6: Slow Binding Inhibitors

6: Slow Binding Inhibitors

Carmela GIGLIONE, Laboratory Head, PhD, Université Paris-Saclay, Paris

Isabelle ARTAUD, Research Director, PhD, French National Centre for Scientific Research, Paris, CNRS, Chemistry and Biology Interdisciplinar Centre paris Descartes University france

A unique peptide deformylase platform to rationally design and challenge novel active compounds

Sonia Fieulaine's research works Université Paris-Saclay, Paris and other places